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Tag: Bioactive Compound Synthesis and Design

New LsrK ligands as AI-2 Quorum Sensing Interfering Compounds Against Biofilm Formation

13 Aprile 2023 admin Publication

Milli G., Pellegrini A., Listro R., Fasolini M., Pagano K., Ragona L., Pietrocola G., Linciano P., Collina S. (2024) Journal of Medicinal Chemistry DOI: 10.1021/acs.jmedchem.4c01266 ABSTRACT:

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Biophysical Assays for Investigating Modulators of Macromolecular Complexes: An OverviewContinuous-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds

13 Aprile 2023 admin Publication

Garbagnoli M., Linciano P., Listro R., Rossino G., Vasile F., Collina S. (2024) ACS Omega 9(16), 17691–17705 DOI: 10.1021/acsomega.4c01309 ABSTRACT: Drug discovery is a lengthy and intricate

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A Green Heck Reaction Protocol towards Trisubstituted Alkenes, Versatile Pharmaceutical Intermediates.

13 Aprile 2023 admin Publication

Rossino G., Marrubini G., Brindisi M., Granje M., Linciano P., Rossi D., Collina, S. (2024) Front. Chem. 12, 1431382 DOI: 10.3389/fchem.2024.1431382 ABSTRACT: The Heck reaction is

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Biocatalysis: A Smart and Green Tool for the Preparation of Chiral Drugs

11 Ottobre 2022 admin Publication

Rossino, G., Robescu, M. S., Licastro, E., Tedesco, C., Martello, I., Maffei, L., Vincenti, G., Bavaro, T., Collina, S. (2022) Chirality, 34(11), pp. 1403–1418.  DOI: 10.1002/chir.23498 ABSTRACT:

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