{"id":453,"date":"2020-11-16T17:13:22","date_gmt":"2020-11-16T16:13:22","guid":{"rendered":"https:\/\/labmedchem.unipv.it\/?page_id=453"},"modified":"2020-11-16T17:13:22","modified_gmt":"2020-11-16T16:13:22","slug":"list-of-publication-of-linciano-pasquale","status":"publish","type":"page","link":"https:\/\/labmedchem.unipv.it\/index.php\/list-of-publication-of-linciano-pasquale\/","title":{"rendered":"List of Publication of Linciano Pasquale"},"content":{"rendered":"\n<p>(1) \u00a0\u00a0\u00a0\u00a0 Ammazzalorso, A.; D\u2019Angelo, A.; Giancristofaro, A.; De Filippis, B.; Di Matteo, M.; Fantacuzzi, M.; Giampietro, L.;\u00a0<strong>Linciano, P.<\/strong>; Maccallini, C.; Amoroso, R. Fibrate-Derived N-(Methylsulfonyl)Amides with Antagonistic Properties on PPAR\u03b1.\u00a0<em>Eur. J. Med. Chem.<\/em>\u00a0<strong>2012<\/strong>, 58, 317\u2013322.\u00a0<a href=\"https:\/\/doi.org\/10.1016\/j.ejmech.2012.10.019\">https:\/\/doi.org\/10.1016\/j.ejmech.2012.10.019<\/a>. <\/p>\n\n\n\n<p>(2) \u00a0\u00a0\u00a0\u00a0 Giampietro, L.; D\u2019Angelo, A.; Giancristofaro, A.; Ammazzalorso, A.; De Filippis, B.; Fantacuzzi, M.;\u00a0<strong>Linciano, P.<\/strong>; Maccallini, C.; Amoroso, R. Synthesis and Structure-Activity Relationships of Fibrate-Based Analogues inside PPARs.\u00a0<em>Bioorganic Med. Chem. Lett.<\/em>\u00a0<strong>2012<\/strong>, 22 (24), 7662\u20137666.\u00a0<a href=\"https:\/\/doi.org\/10.1016\/j.bmcl.2012.09.111\">https:\/\/doi.org\/10.1016\/j.bmcl.2012.09.111<\/a>. <\/p>\n\n\n\n<p>(3) \u00a0\u00a0\u00a0\u00a0\u00a0<strong>Linciano, P.<\/strong>; Pizzetti, M.; Porcheddu, A. Use of Primary Amines for the Selective N-Alkylation of Anilines by a Reusab- Le Heterogeneous Catalyst.\u00a0<em>Synlett<\/em>\u00a0<strong>2013<\/strong>, 24, 2249\u20132254.\u00a0<a href=\"https:\/\/doi.org\/10.1055\/s-0033-1339667\">https:\/\/doi.org\/10.1055\/s-0033-1339667<\/a>.<\/p>\n\n\n\n<p>(4) \u00a0\u00a0\u00a0\u00a0 Giampietro, L.; D\u2019Angelo, A.; Giancristofaro, A.; Ammazzalorso, A.; De Filippis, B.; Di Matteo, M.; Fantacuzzi, M.;\u00a0<strong>Linciano, P.<\/strong>; Maccallini, C.; Amoroso, R. Effect of Stilbene and Chalcone Scaffolds Incorporation in Clofibric Acid on PPAR\u03b1 Agonistic Activity.\u00a0<em>Med. Chem.<\/em>\u00a0<strong>2014<\/strong>, 10 (1), 59\u201365. <\/p>\n\n\n\n<p>(5) \u00a0\u00a0\u00a0\u00a0 De Filippis, B.;\u00a0<strong>Linciano, P.<\/strong>; Ammazzalorso, A.; Di Giovanni, C.; Fantacuzzi, M.; Giampietro, L.; Laghezza, A.; Maccallini, C.; Tortorella, P.; Lavecchia, A.; et al. Structural Development Studies of PPARs Ligands Based on Tyrosine Scaffold.\u00a0<em>Eur. J. Med. Chem.<\/em>\u00a0<strong>2015<\/strong>, 89, 817\u2013825.\u00a0<a href=\"https:\/\/doi.org\/10.1016\/j.ejmech.2014.10.083\">https:\/\/doi.org\/10.1016\/j.ejmech.2014.10.083<\/a>. <\/p>\n\n\n\n<p>(6) \u00a0\u00a0\u00a0\u00a0 Quotadamo, A.;\u00a0<strong>Linciano, P.<\/strong>; Davoli, P.; Tondi, D.; Costi, M. P.; Venturelli, A. An Improved Synthesis of CENTA, a Chromogenic Substrate for \u03b2-Lactamases.\u00a0<em>Synlett<\/em>\u00a0<strong>2016<\/strong>, 27 (17), 2447\u20132450.\u00a0<a href=\"https:\/\/doi.org\/10.1055\/s-0035-1562454\">https:\/\/doi.org\/10.1055\/s-0035-1562454<\/a>. <\/p>\n\n\n\n<p>(7) \u00a0\u00a0\u00a0\u00a0\u00a0<strong>Linciano, P.<\/strong>; Ammazzalorso, A.; De Filippis, B.; Fantacuzzi, M.; Giampietro, L.; Maccallini, C.; Amoroso, R. Geometric Isomerism of an Acetamidino Derivative Determined by NMR Investigations.\u00a0<em>ChemistrySelect<\/em>\u00a0<strong>2017<\/strong>, 2 (30), 9706\u20139710. \u00a0<a href=\"https:\/\/doi.org\/10.1002\/slct.201701646\">https:\/\/doi.org\/10.1002\/slct.201701646<\/a>. <\/p>\n\n\n\n<p>(8) \u00a0\u00a0\u00a0\u00a0 Borsari, C.; Santarem, N.; Torrado, J.; Ol\u00edas, A. I.; Corral, M. J.; Baptista, C.; Gul, S.; Wolf, M.; Kuzikov, M.; Ellinger, B.;\u00a0<strong>Linciano, P.<\/strong>; et al. Methoxylated 2\u2019-Hydroxychalcones as Antiparasitic Hit Compounds.\u00a0<em>Eur. J. Med.\u00a0Chem.<\/em>\u00a0<strong>2017<\/strong>, 126, 1129\u20131135.\u00a0<a href=\"https:\/\/doi.org\/10.1016\/j.ejmech.2016.12.017\">https:\/\/doi.org\/10.1016\/j.ejmech.2016.12.017<\/a>. <\/p>\n\n\n\n<p>(9) \u00a0\u00a0\u00a0\u00a0\u00a0<strong>Linciano, P.<\/strong>; Dawson, A.; P\u00f6hner, I.; Costa, D. M.; Sa, M. S.; Cordeiro-Da-Silva, A.; Luciani, R.; Gul, S.; Witt, G.; Ellinger, B.; et al. Exploiting the 2\u2011Amino-1,3,4-Thiadiazole Scaffold to Inhibit Trypanosoma Brucei Pteridine Reductase in Support of Early-Stage Drug Discovery.\u00a0<em>ACS Omega<\/em>\u00a0<strong>2017<\/strong>, 2 (9), 5666\u20135683.\u00a0<a href=\"https:\/\/doi.org\/10.1021\/acsomega.7b00473\">https:\/\/doi.org\/10.1021\/acsomega.7b00473<\/a>. <\/p>\n\n\n\n<p>(10) \u00a0\u00a0\u00a0<strong>Linciano, P.<\/strong>; Moraes, C. B.; Alcantara, L. M.; Franco, C. H.; Pascoalino, B.; Freitas-Junior, L. H.; Macedo, S.; Santarem, N.; Cordeiro-da-Silva, A.; Gul, S.; et al. Aryl Thiosemicarbazones for the Treatment of Trypanosomatidic Infections.\u00a0<em>Eur. J. Med. Chem.<\/em>\u00a0<strong>2018<\/strong>, 146, 423\u2013434.\u00a0<a href=\"https:\/\/doi.org\/10.1016\/j.ejmech.2018.01.043\">https:\/\/doi.org\/10.1016\/j.ejmech.2018.01.043<\/a>. <\/p>\n\n\n\n<p>(11) \u00a0\u00a0 Celenza, G.; Vicario, M.; Bellio, P.;\u00a0<strong>Linciano, P.<\/strong>; Perilli, M.; Oliver, A.; Blazquez, J.; Cendron, L.; Tondi, D. Phenylboronic Acid Derivatives as Validated Leads Active in Clinical Strains Overexpressing KPC-2: A Step against Bacterial Resistance.\u00a0<em>ChemMedChem<\/em>\u00a0<strong>2018<\/strong>.\u00a0<a href=\"https:\/\/doi.org\/10.1002\/cmdc.201700788\">https:\/\/doi.org\/10.1002\/cmdc.201700788<\/a>.<\/p>\n\n\n\n<p>(12) \u00a0\u00a0 Klein, R.;\u00a0<strong>Linciano, P.<\/strong>; Celenza, G.; Bellio, P.; Papaioannou, S.; Blazquez, J.; Cendron, L.; Brenk, R.; Tondi, D. In Silico Identification and Experimental Validation of Hits Active against KPC-2 \u03b2-Lactamase.\u00a0<em>PLoS One<\/em>\u00a0<strong>2018<\/strong>, 13 (11), 1\u201322.\u00a0<a href=\"https:\/\/doi.org\/10.1371\/journal.pone.0203241\">https:\/\/doi.org\/10.1371\/journal.pone.0203241<\/a>.<\/p>\n\n\n\n<p>(13) \u00a0\u00a0 Franchini, S.; Sorbi, C.;\u00a0<strong>Linciano, P.<\/strong>; Brasili, L.; Tait, A. Effect of the Rigidification of Propranolol, a Mixed Beta-Adrenoceptor and 5-HT1AR Antagonist.\u00a0<em>Pharmazie<\/em>\u00a0<strong>2019<\/strong>, 74 (3), 131\u2013135.\u00a0<a href=\"https:\/\/doi.org\/10.1691\/ph.2019.8878\">https:\/\/doi.org\/10.1691\/ph.2019.8878<\/a>. <\/p>\n\n\n\n<p>(14) \u00a0\u00a0 Landi, G.;\u00a0<strong>Linciano, P.<\/strong>; Borsari, C.; Bertolacini, C. P.; Moraes, C. B.; Cordeiro-Da-Silva, A.; Gul, S.; Witt, G.; Kuzikov, M.; Costi, M. P.; et al. Structural Insights into the Development of Cycloguanil Derivatives as Trypanosoma Brucei Pteridine-Reductase-1 Inhibitors.\u00a0<em>ACS Infect. Dis.<\/em>\u00a0<strong>2019<\/strong>, 5, 1105\u20131114.\u00a0<a href=\"https:\/\/doi.org\/10.1021\/acsinfecdis.8b00358\">https:\/\/doi.org\/10.1021\/acsinfecdis.8b00358<\/a>. <\/p>\n\n\n\n<p>(15) \u00a0\u00a0 Citti, C.;\u00a0<strong>Linciano, P.<\/strong>; Panseri, S.; Vezzalini, F.; Forni, F.; Vandelli, M. A.; Cannazza, G. Cannabinoid Profiling of Hemp Seed Oil by Liquid Chromatography Coupled to High-Resolution Mass Spectrometry.\u00a0<em>Front. Plant Sci.<\/em>\u00a0<strong>2019<\/strong>, 10 (February), 1\u201317.\u00a0<a href=\"https:\/\/doi.org\/10.3389\/fpls.2019.00120\">https:\/\/doi.org\/10.3389\/fpls.2019.00120<\/a>. <\/p>\n\n\n\n<p>(16) \u00a0\u00a0 Spyrakis, F.; Bellio, P.; Quotadamo, A.;\u00a0<strong>Linciano, P.<\/strong>; Benedetti, P.; D\u2019Arrigo, G.; Baroni, M.; Cendron, L.; Celenza, G.; Tondi, D. First Virtual Screening and Experimental Validation of Inhibitors Targeting GES-5 Carbapenemase.\u00a0<em>J. Comput. Aided. Mol. Des.<\/em>\u00a0<strong>2019<\/strong>, 33 (2), 295\u2013305.\u00a0<a href=\"https:\/\/doi.org\/10.1007\/s10822-018-0182-2\">https:\/\/doi.org\/10.1007\/s10822-018-0182-2<\/a>. <\/p>\n\n\n\n<p>(17) \u00a0\u00a0 Moraes, C. B.; Witt, G.; Kuzikov, M.; Ellinger, B.; Calogeropoulou, T.; Prousis, K. C.; Mangani, S.; Di Pisa, F.; Landi, G.; Iacono, L. Dello;\u00a0<strong>Linciano, P.<\/strong>\u00a0et al. Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform.\u00a0<em>SLAS Discov. Adv. Life Sci. R&amp;D<\/em>\u00a0<strong>2019<\/strong>, 24 (3), 346\u2013361.\u00a0<a href=\"https:\/\/doi.org\/10.1177\/2472555218823171\">https:\/\/doi.org\/10.1177\/2472555218823171<\/a>.<\/p>\n\n\n\n<p>(18) \u00a0\u00a0 Quotadamo, A.;\u00a0<strong>Linciano, P.<\/strong>; Costi, M. P.; Venturelli, A. Optimization of N \u2010alkylation in the Synthesis of Methotrexate and Pteridine\u2010based Derivatives Under Microwave\u2010Irradiation.\u00a0<em>ChemistrySelect<\/em>\u00a0<strong>2019<\/strong>, 4 (15), 4429\u20134433.\u00a0<a href=\"https:\/\/doi.org\/10.1002\/slct.201900721\">https:\/\/doi.org\/10.1002\/slct.201900721<\/a>. <\/p>\n\n\n\n<p>(19) \u00a0\u00a0\u00a0<strong>Linciano, P.*<\/strong>; Pozzi, C.; Iacono, L. Dello; Di Pisa, F.; Landi, G.; Bonucci, A.; Gul, S.; Kuzikov, M.; Ellinger, B.; Witt, G.; et al. Enhancement of Benzothiazoles as Pteridine Reductase-1 Inhibitors for the Treatment of Trypanosomatidic Infections.\u00a0<em>J. Med. Chem.<\/em>\u00a0<strong>2019<\/strong>, 62 (8), 3989\u20134012.\u00a0<a href=\"https:\/\/doi.org\/10.1021\/acs.jmedchem.8b02021\">https:\/\/doi.org\/10.1021\/acs.jmedchem.8b02021<\/a>. <\/p>\n\n\n\n<p>(20) \u00a0\u00a0 Franchini, S.; Sorbi, C.;\u00a0<strong>Linciano, P.<\/strong>; Carnevale, G.; Tait, A.; Ronsisvalle, S.; Buccioni, M.; Del Bello, F.; Cilia, A.; Pirona, L.; et al. 1,3-Dioxane as a Scaffold for Potent and Selective 5-HT 1A R Agonist with in-Vivo Anxiolytic, Anti-Depressant and Anti-Nociceptive Activity.\u00a0<em>Eur. J. Med. Chem.<\/em>\u00a0<strong>2019<\/strong>, 176, 310\u2013325.\u00a0<a href=\"https:\/\/doi.org\/10.1016\/j.ejmech.2019.05.024\">https:\/\/doi.org\/10.1016\/j.ejmech.2019.05.024<\/a>. <\/p>\n\n\n\n<p>(21) \u00a0\u00a0\u00a0<strong>Linciano, P.<\/strong>; Cendron, L.; Gianquinto, E.; Spyrakis, F.; Tondi, D. Ten Years with New Delhi Metallo-\u03b2-Lactamase-1 (NDM-1): From Structural Insights to Inhibitor Design.\u00a0<em>ACS Infect. Dis.<\/em>\u00a0<strong>2019<\/strong>, 5 (1), 9\u201334.\u00a0<a href=\"https:\/\/doi.org\/10.1021\/acsinfecdis.8b00247\">https:\/\/doi.org\/10.1021\/acsinfecdis.8b00247<\/a>. <\/p>\n\n\n\n<p>(22) \u00a0\u00a0 Vanossi, D.; Casell, M.; Pavesi, G.; Borsari, C.;\u00a0<strong>Linciano, P.<\/strong>; Costi, M. P.; Ponterini, G. Excited-State Intramolecular Proton Transfer in a Bioactive Flavonoid Provides Fluorescence Observables for Recognizing Its Engagement with Target Proteins.\u00a0<em>Photochem. Photobiol. Sci.<\/em>\u00a0<strong>2019<\/strong>.\u00a0<a href=\"https:\/\/doi.org\/10.5860\/choice.51-2070\">https:\/\/doi.org\/10.5860\/choice.51-2070<\/a>. <\/p>\n\n\n\n<p>(23) \u00a0\u00a0 Citti, C.;\u00a0<strong>Linciano, P. (co-first)<\/strong>; Forni, F.; Vandelli, M. A.; Gigli, G.; Lagan\u00e0, A.; Cannazza, G. Analysis of Impurities of Cannabidiol from Hemp. Isolation, Characterization and Synthesis of Cannabidibutol, the Novel Cannabidiol Butyl Analog.\u00a0<em>J. Pharm. Biomed. Anal.<\/em>\u00a0<strong>2019<\/strong>.\u00a0<a href=\"https:\/\/doi.org\/10.1016\/j.jpba.2019.06.049\">https:\/\/doi.org\/10.1016\/j.jpba.2019.06.049<\/a>. <\/p>\n\n\n\n<p>(24)\u00a0\u00a0\u00a0\u00a0<strong>Linciano, P.;<\/strong>\u00a0De Filippis, B.; Ammazzalorso, A.; Amoia, P.; Fantacuzzi, M.; Giampietro, L.; Maccallini, C.; Petit, C.; Amoroso, R. Druggability Profile of Stilbene-Derived PPAR Agonists\u202f: Determination of Physicochemical Properties and PAMPA Druggability Profile of Stilbene-Derived PPAR Agonists\u202f: Determination of Physicochemical Properties and PAMPA Study.\u00a0<em>Medchemcomm<\/em>\u00a0<strong>2019<\/strong>,\u00a0<a href=\"https:\/\/doi.org\/10.1039\/C9MD00286C\">https:\/\/doi.org\/10.1039\/C9MD00286C<\/a>. <\/p>\n\n\n\n<p>(25) \u00a0\u00a0 Borsari, C.; Jim\u00e9nez-ant\u00f3n, M. D.; Eick, J.; Bifeld, E.; Jos\u00e9, J.; Ol\u00edas-molero, A. I.; Corral, M. J.; Santarem, N.; Severi, L.; Gul, S.;\u00a0<strong>Linciano, P.<\/strong>\u00a0et al. Discovery of a Benzothiophene-Flavonol Halting Miltefosine and Antimonial Drug Resistance in Leishmania Parasites through the Application of Medicinal Chemistry, Screening and Genomics.\u00a0<em>Eur. J. Med. Chem.<\/em>\u00a0<strong>2019<\/strong>, 111676,\u00a0<a href=\"https:\/\/doi.org\/10.1016\/j.ejmech.2019.111676\">https:\/\/doi.org\/10.1016\/j.ejmech.2019.111676<\/a>. <\/p>\n\n\n\n<p>(26) \u00a0\u00a0 Citti, C.;\u00a0<strong>Linciano, P. (co-first);<\/strong>\u00a0Forni, F.; Vandelli, M. A.; Gigli, G.; Lagan\u00e0, A.; Cannazza, G. Chemical and Spectroscopic Characterization Data of \u2018Cannabidibutol\u2019, a Novel Cannabidiol Butyl Analog.\u00a0<em>Data Br.<\/em>\u00a0<strong>2019<\/strong>, 104463,\u00a0<a href=\"https:\/\/doi.org\/10.1016\/j.dib.2019.104463\">https:\/\/doi.org\/10.1016\/j.dib.2019.104463<\/a>. <\/p>\n\n\n\n<p>(27)\u00a0\u00a0\u00a0\u00a0<strong>Linciano, P.<\/strong>; Vicario, M.; Kekez, I.; Bellio, P.; Celenza, G.; Martin-Blecua, I.; Blazquez, J.; Cendron, L.; Tondi, D. Phenyl boronic acids probing molecular recognition 3 against class A and class C \u03b2-lactamases.\u00a0<em>Antibiotics,\u00a0<\/em><strong>2019<\/strong><em>,\u00a0<\/em>8 (4), art. no. 171. DOI: 10.3390\/antibiotics804017.<\/p>\n\n\n\n<p>(28)\u00a0\u00a0\u00a0\u00a0<strong>Linciano, P.<\/strong>; Cullia, G.; Borsari, C.; Santucci, M.; Ferrari, S.; Witt, G.; Gul, S.; Santarem, N.; Cordeiro da Silva, A.; et al.\u00a0<em>Trypanosoma<\/em>\u00a0<em>brucei<\/em>\u00a0screening fishes out a 2,4-diaminopyrimidine scaffold targeting pteridine reductase 1 from the LIBRA compound library HTS campaign.\u00a0<em>Eur. J. Med. Chem<\/em>.\u00a0<strong>2019<\/strong>, 189, art. No. 112047.DOI: 10.1016\/j.ejmech.2020.112047.<\/p>\n\n\n\n<p>(29)\u00a0\u00a0\u00a0 Pacifico, S.; Santucci, M.; Luciani, R.; Saxena P.;\u00a0<strong>Linciano, P.;<\/strong>\u00a0Ponterini, G.; D\u2019Arca, D.; Marverti, G.; Guerrini, R.; Costi, M. P. Cyclic peptides acting as allosteric inhibitors of human thymidylate synthase and cancer cell growth.\u00a0<em>Molecules.\u00a0<\/em><strong>2019<\/strong><em>,\u00a0<\/em>24 (19), art. no. 3493<em>.\u00a0<\/em>DOI: 10.3390\/molecules24193493.<\/p>\n\n\n\n<p>(30)\u00a0\u00a0\u00a0\u00a0<strong>Linciano, P.;<\/strong>\u00a0Citti, C.; Luongo, L.; Belardo, C.; Vandelli, M.A.; Forni, F.; Gigli, G.; Lagan\u00e0, A.; Montone, C; Cannazza, C.; Isolation of a high affinity cannabinoid for human CB1 receptor from a medicinal cannabis variety: tetrahydrocannabutol, the butyl analog of tetrahydrocannabinol.\u00a0<em>Journal of Natural Products.\u00a0<\/em><strong>2019<\/strong>. 175, art. no. 112752. DOI: 10.1016\/j.jpba.2019.06.049. <\/p>\n\n\n\n<p>(31)\u00a0\u00a0\u00a0 Citti, C.,\u00a0<strong>Linciano, P. (co-first),<\/strong>\u00a0Russo, F., Luongo, L., Iannotta, M., Maione, S., Lagan\u00e0, A., Capriotti, A.L., Forni, F., Vandelli, M.A., Gigli, G., Cannazza, G. A novel phytocannabinoid isolated from Cannabis sativa L. with an in vivo cannabimimetic activity higher than \u03949-tetrahydrocannabinol: \u03949-Tetrahydrocannabiphorol.\u00a0<em>Scientific Reports<\/em>.\u00a0<strong>2019<\/strong>, 9 (1), art. no. 20335. DOI: 10.1038\/s41598-019-56785-1. <\/p>\n\n\n\n<p>(32)\u00a0\u00a0\u00a0\u00a0<strong>Linciano, P.,<\/strong>\u00a0Gianquinto, E., Montanari, M., Maso, L., Bellio, P., Cebri\u00e1n-Sastre, E., Celenza, G., Bl\u00e1zquez, J., Cendron, L., Spyrakis, F., Tondi, D. 4-amino-1,2,4-triazole-3-thione as a promising scaffold for the inhibition of serine and metallo-\u03b2-lactamases.\u00a0<em>Pharmaceuticals<\/em>.\u00a0<strong>2020<\/strong>, 13 (3), art. no. 52. DOI: 10.3390\/ph13030052. <\/p>\n\n\n\n<p>(33)\u00a0\u00a0\u00a0 Citti, C.,\u00a0<strong>Linciano, P.,<\/strong>\u00a0Cannazza, G. Is cannabidiol a scheduled controlled substance? Origin makes the difference. Drug Discovery Today. 2020, 25 (4), pp. 628-632. DOI: 10.1016\/j.drudis.2020.02.001. <\/p>\n\n\n\n<p>(34)\u00a0\u00a0\u00a0 Franchini, S<strong>., Linciano, P<\/strong>., Puja, G., Tait, A., Borsari, C., Denora, N., Iacobazzi, R.M., Brasili, L., Sorbi, C. Novel Dithiolane-Based Ligands Combining Sigma and NMDA Receptor Interactions as Potential Neuroprotective Agents.\u00a0<em>ACS Medicinal Chemistry Letters<\/em>.\u00a0<strong>2020<\/strong>, 11 (5), pp. 1028-1034. DOI: 10.1021\/acsmedchemlett.0c00129. <\/p>\n\n\n\n<p>(35)\u00a0\u00a0\u00a0 Landi, G.,\u00a0<strong>Linciano, P.,<\/strong>\u00a0Tassone, G., Costi, M.P., Mangani, S., Pozzi, C. High-resolution crystal structure of Trypanosoma brucei pteridine reductase 1 in complex with an innovative tricyclic-based inhibitor.\u00a0<em>Acta Crystallographica Section D: Structural Biology<\/em>.\u00a0<strong>2020<\/strong>, 76, pp. 558-564. DOI: 10.1107\/S2059798320004891. <\/p>\n\n\n\n<p>(36)\u00a0\u00a0\u00a0\u00a0<strong>Linciano, P.,<\/strong>\u00a0Rossino, G., Listro, R., Rossi, D., Collina, S. The sigma-1 receptor antagonists, promising players in fighting neuropathic pain.\u00a0<em>Pharmaceutical Patent Analysis<\/em>.\u00a0<strong>2020<\/strong>, DOI: 10.4155\/ppa-2020-0007. <\/p>\n\n\n\n<p>(37)\u00a0\u00a0\u00a0 Citti, C., Russo, F.,\u00a0<strong>Linciano, P<\/strong>., Strallhofer, S.S., Tolomeo, F., Forni, F., Vandelli, M.A., Gigli, G., Cannazza, G. Origin of D9-Tetrahydrocannabinol Impurity in Synthetic Cannabidiol.\u00a0<em>Cannabis and Cannabinoids Research<\/em>.\u00a0<strong>2020<\/strong>, DOI: 10.1089\/can.2020.0021. <\/p>\n\n\n\n<p>(38)\u00a0\u00a0\u00a0 Rossino, G., Rui, M., Pozzetti, L., Schepmann, D., W\u00fcnsch, B., Zambieri, D, Pellavio, G., Laforenza, U., Rinaldi, S., Colombo, G., Morelli, L.,\u00a0<strong>Linciano, P.,<\/strong>\u00a0Rossi, D., Collina, S.\u00a0<a href=\"https:\/\/pasqualelinciano.wordpress.com\/2020\/10\/17\/setup-and-validation-of-a-reliable-docking-protocol-for-the-development-of-neuroprotective-agents-by-targeting-the-sigma-1-receptor-s1r\/\">Setup and Validation of a Reliable Docking Protocol for the Development of Neuroprotective Agents by Targeting the Sigma-1 Receptor (S1R).\u00a0<\/a>Int. J. Mol. Sci.\u00a0<strong>2020<\/strong>.\u00a0<em>Just accepted<\/em>. <\/p>\n","protected":false},"excerpt":{"rendered":"<p>(1) \u00a0\u00a0\u00a0\u00a0 Ammazzalorso, A.; D\u2019Angelo, A.; Giancristofaro, A.; De Filippis, B.; Di Matteo, M.; Fantacuzzi, M.; Giampietro, L.;\u00a0Linciano, P.; Maccallini, C.; Amoroso, R. Fibrate-Derived N-(Methylsulfonyl)Amides<\/p>\n","protected":false},"author":1,"featured_media":0,"parent":0,"menu_order":0,"comment_status":"closed","ping_status":"closed","template":"","meta":[],"_links":{"self":[{"href":"https:\/\/labmedchem.unipv.it\/index.php\/wp-json\/wp\/v2\/pages\/453"}],"collection":[{"href":"https:\/\/labmedchem.unipv.it\/index.php\/wp-json\/wp\/v2\/pages"}],"about":[{"href":"https:\/\/labmedchem.unipv.it\/index.php\/wp-json\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"https:\/\/labmedchem.unipv.it\/index.php\/wp-json\/wp\/v2\/users\/1"}],"replies":[{"embeddable":true,"href":"https:\/\/labmedchem.unipv.it\/index.php\/wp-json\/wp\/v2\/comments?post=453"}],"version-history":[{"count":1,"href":"https:\/\/labmedchem.unipv.it\/index.php\/wp-json\/wp\/v2\/pages\/453\/revisions"}],"predecessor-version":[{"id":455,"href":"https:\/\/labmedchem.unipv.it\/index.php\/wp-json\/wp\/v2\/pages\/453\/revisions\/455"}],"wp:attachment":[{"href":"https:\/\/labmedchem.unipv.it\/index.php\/wp-json\/wp\/v2\/media?parent=453"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}