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Tag: Bioactive Compound Synthesis and Design

From Nature to Synthetic Compounds: Novel 1(N),2,3 Trisubstituted-5-oxopyrrolidines Targeting Multiple Myeloma Cells

27 Ottobre 2022 admin Publication

Listro, R., Malacrida, A., Ambrosio, F.A., Rossino, G., Di Giacomo, M., Cavalloro, V., Garbagnoli, M., Linciano, P., Rossi, D., Cavaletti, G., Costa, G., Alcaro, S.,

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Biocatalysis: A Smart and Green Tool for the Preparation of Chiral Drugs

11 Ottobre 2022 admin Publication

Rossino, G., Robescu, M. S., Licastro, E., Tedesco, C., Martello, I., Maffei, L., Vincenti, G., Bavaro, T., Collina, S. (2022) Chirality, 34(11), pp. 1403–1418.  DOI: 10.1002/chir.23498 ABSTRACT:

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Synthesis and Characterization of a “Clickable” PBR28 TSPO-Selective Ligand Derivative Suitable for the Functionalization of Biodegradable Polymer Nanoparticles.

11 Ottobre 2022 admin Publication

Auriemma, R., Sponchioni, M., Capasso Palmiero, U., Rossino, G., Rossetti, A., Marsala, A., Collina, S., Sacchetti, A., Moscatelli, D., Peviani, M. (2021) Nanomaterials, 11, 1693. DOI: 10.3390/nano11071693

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Effects of endocrine active contaminating pesticides on RACK1 expression and immunological consequences in THP-1 cells

11 Ottobre 2022 admin Publication

Maddalon, A., Masi, M., Iulini, M., Linciano, P., Galbiati, V., Marinovich, M., Racchi, M., Buoso, E., Corsini, E. (2022) Environmental Toxicology and Pharmacology, 95, art.

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Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1.

11 Ottobre 2022 admin Publication

Pöhner, I., Quotadamo, A., Panecka-Hofman, J., Luciani, R., Santucci, M., Linciano, P., Landi, G., Di Pisa, F., Dello Iacono, L., Pozzi, C., Mangani, S., Gul,

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